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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5622 | BAY-218 | AHR antagonist 1 | AhR , Aryl Hydrocarbon Receptor |
BAY-218 (AHR antagonist 1) is an aryl hydrocarbon receptor (AHR) antagonist , has an IC50 of 39.9 nM in human cell line. | |||
T9822 | WAY-605471 | AhR | |
WAY-605471 is a AHR antagonist with IC50 of 0.5 - 1 μM. | |||
T5541 | PDM11 | 1-[2-(4-Chloro-phenyl)-vinyl]-3,5-diMeth,PDM 11 | AhR |
PDM11 (1-[2-(4-Chloro-phenyl)-vinyl]-3,5-diMeth) is an antagonist of aryl hydrocarbon receptor (AhR) | |||
T10272 | AHR antagonist 5 | Others | |
AHR antagonist 5 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist(example 39; IC50 < 0.5 μΜ). It significantly inhibits tumor growth combined with checkpoint inhibitor anti-PD-1. | |||
T63389 | AHR antagonist 5 hemimaleate | ||
AHR antagonist 5 hemimaleate is a potent antagonist (IC50 < 0.5 μM) of the orally active aryl hydrocarbon receptor (AHR). aHR antagonist 5 hemimaleate in combination with the detection site inhibitor anti-PD-1 exhibited ... | |||
T72056 | KYN-101 | ||
KYN-101 is a potent, selective synthetic antagonist of aryl hydrocarbon receptor (AHR) with IC50 of 22 nM in human HepG2 DRE-luciferase reporter assay and 23 nM in murine Hepa1 Cyp-luc assay.KYN-101 reverses IDO/TDO-medi... |